Ulwakhiwo lweMolekyuli:
I-cytisine yi-alkaloid yendalo ifumaneka kwiintlobo ezahlukeneyo zezityalo, ezinje ngeCytisus Cradenum naseLaburnium AsanaDroides. Isetyenziselwe iminyaka emininzi njengoncedo lokutshaya ngenxa yokufana ne-nicotine.Umsebenzi ophambili we-cytisine njengogqirha we-agoninic acetycholic (i-nachrs). Ezi ndawo zikhutshiweyo zifumaneka kwingqondo, ngokukodwa kwiindawo ezibandakanyeka kwiziyobisi, kwaye zinoxanduva lokucamngca ngeziphumo ezinomvuzo zeNicotine. Ngokubopha kunye nokwenza ezi zinto zikhutshiweyo, i-cytisine inceda ukunciphisa iminqweno ye-nicotine kunye neempawu zokurhoxa ngexesha lokutshaya.cytisine zibonakalisiwe ukuba lunyango olusebenzayo lwe-nicico kwizifundo ezahlukeneyo zeklinikhi. Inganceda ukuphucula amaxabiso okuyeka kwaye kuncitshiswe ubungqingqwa beempawu zokurhoxa, zenze ukuba kuluncedo kwiinkqubo zokutshaya ukutshaya.
Kubalulekile ukuba uqaphele ukuba i-cytisine inokuba neziphumo ebezingalindelekanga, ezinjenge-nausea, ukugabha, kunye nokuphazamiseka okulala. Njengalo naluphi na unyango, kufuneka lusetyenziswe njengoko kuyalelwe kwaye phantsi kweliso lezempilo yezempilo. Ukuba ucinga usebenzisa i-cytisine njengoncedo lokutshaya, ndicebisa ukuba ndithethe nodokotela ukuba icebiso kunye nesikhokelo.
Into | Ukucaciswa | |
I-Assay (i-HPPC) | ||
I-cytisine: | ≥98% | |
Umgangatho: | I-CP2010 | |
I-procisochemical | ||
Imbonakalo: | I-rystalline ye-crystalline | |
I-Odor: | I-Oder ye-Oder | |
Unizi lolwapho kuyiwa khona: | I-50-60g / 100ml | |
UMesh: | I-95% ye-80mesh | |
Intsimbi enzima: | ≤10ppm | |
Njenge: | ≤2ppm | |
I-PB: | ≤2ppm | |
Ilahleko yokomisa: | ≤1% | |
Intsalela yentsalela: | ≤0.1% | |
Intsalela yeSolvent: | ≤3000ppm |